Synthesis of ?-substituted indolylacetamide using acetonitriles as acetamide enolate equivalents through O-transfer reactions
نویسندگان
چکیده
The combination of hemiaminals and acetonitriles unlocks the novel reactivities, such as that an O-transfer reagent a masked amide enolate, enabling synthesis ?-substituted indolylacetamides through alkylation/O-transfer reaction.
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ژورنال
عنوان ژورنال: Chemical Communications
سال: 2021
ISSN: ['1359-7345', '1364-548X']
DOI: https://doi.org/10.1039/d1cc02821a